912369-50-7 4-Piperazinylphenylboronic Acid, Pinacol Ester

912369-50-7 4-Piperazinylphenylboronic Acid, Pinacol Ester

1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine Basic information 1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine Chemical Properties Safety Information MSDS Information 1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine Usage And...
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Product Details

1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine Basic information

Product Name:

1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine

Synonyms:

1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine;3-Hydroxy-2,3-diMethylbutan-2-yl    hydrogen (2-(piperazin-1-yl)phenyl)boronate;1-[4-(tetraMethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperazine;4-Piperazinylphenylboronic acid

CAS:

912369-50-7

MF:

C16H25BN2O2

MW:

288.1929

EINECS:

 

Product Categories:

 

Mol File:

912369-50-7.mol

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1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine Chemical Properties

Density:

1.08g/cm3

Boiling   Point:

432.7ºC at 760 mmHg

Flash    Point:

215.5ºC

Refractiv Index:

1.541


Safety Information


MSDS Information


1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine Usage And Synthesis

Uses

suzuki reaction

Intermediate as

1062368-24-4 LDN-193189,1432597-26-6 LDN-212854 and 1062368-62-0 LDN-193189 HCl

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Synthesis route

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Reference:

WO2006/106326 A1, ; Page/Page column 133 ; WO 2006/106326 A1


1-[4-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-piperazine Preparation Products And Raw materials

 

Upstream information

4-(4-Boc-piperazino)phenylboronic Acid Pinacol Ester;


Downtream information

1-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]piperazine;


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